AR058019A1 - Proceso de preparacion de un derivado de pirrolopirimidina - Google Patents

Proceso de preparacion de un derivado de pirrolopirimidina

Info

Publication number
AR058019A1
AR058019A1 ARP060103390A ARP060103390A AR058019A1 AR 058019 A1 AR058019 A1 AR 058019A1 AR P060103390 A ARP060103390 A AR P060103390A AR P060103390 A ARP060103390 A AR P060103390A AR 058019 A1 AR058019 A1 AR 058019A1
Authority
AR
Argentina
Prior art keywords
pirrolopirimidine
derivative
preparation process
phenyl
ethyl
Prior art date
Application number
ARP060103390A
Other languages
English (en)
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of AR058019A1 publication Critical patent/AR058019A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Reivindicacion 1: Un método para la preparacion de {6-[4-(4-etil-piperazin-1-ilmetil)-fenil-7H-pirrolo-[2,3-d]-pirimidin-4-il]-(R-1-fenil-etil)amina, que tiene la formula (1), la cual comprende reducir la fraccion de amida del compuesto de la formula (2).
ARP060103390A 2005-08-05 2006-08-03 Proceso de preparacion de un derivado de pirrolopirimidina AR058019A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US70607105P 2005-08-05 2005-08-05

Publications (1)

Publication Number Publication Date
AR058019A1 true AR058019A1 (es) 2008-01-23

Family

ID=37198768

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP060103390A AR058019A1 (es) 2005-08-05 2006-08-03 Proceso de preparacion de un derivado de pirrolopirimidina

Country Status (15)

Country Link
US (1) US20080227980A1 (es)
EP (1) EP1919917A2 (es)
JP (1) JP2009503034A (es)
KR (1) KR20080040695A (es)
CN (1) CN101238130A (es)
AR (1) AR058019A1 (es)
AU (1) AU2006277997A1 (es)
BR (1) BRPI0614710A2 (es)
CA (1) CA2617720A1 (es)
GT (1) GT200600349A (es)
MX (1) MX2008001611A (es)
PE (1) PE20070415A1 (es)
RU (1) RU2008108089A (es)
TW (1) TW200726770A (es)
WO (1) WO2007017468A2 (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7955473B2 (en) 2004-12-22 2011-06-07 Akzo Nobel N.V. Process for the production of paper
US20060254464A1 (en) 2005-05-16 2006-11-16 Akzo Nobel N.V. Process for the production of paper
US8273216B2 (en) 2005-12-30 2012-09-25 Akzo Nobel N.V. Process for the production of paper
CA2636954A1 (en) * 2006-01-23 2007-07-26 Novartis Ag Solid forms of a pyrrolopyrimidine derivative and their use as anti-tumor agents
EP2446885B1 (en) 2009-06-26 2017-09-06 Teijin Pharma Limited Therapeutic agent for hypertension or normal high blood pressure
CN102762543B (zh) 2010-02-01 2016-03-09 巴斯夫欧洲公司 用于防除动物害虫的取代的酮型异*唑啉化合物和衍生物
AR083646A1 (es) 2010-10-01 2013-03-13 Basf Se Compuestos de imina, composiciones veterinarias y agricolas que los contienen y su uso en el control de plagas de invertebrados
EP2621897A1 (en) 2010-10-01 2013-08-07 Basf Se Imine compounds
CN110498812B (zh) * 2018-05-17 2021-08-24 上海医药工业研究院 一种艾拉普林的中间体化合物的制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR9609617B1 (pt) * 1995-07-06 2010-07-27 derivados de 7h-pirrol[2,3-d]pirimidina, e composição farmacêutica.
GB0119249D0 (en) * 2001-08-07 2001-10-03 Novartis Ag Organic compounds

Also Published As

Publication number Publication date
US20080227980A1 (en) 2008-09-18
GT200600349A (es) 2007-02-28
EP1919917A2 (en) 2008-05-14
AU2006277997A1 (en) 2007-02-15
TW200726770A (en) 2007-07-16
CN101238130A (zh) 2008-08-06
BRPI0614710A2 (pt) 2011-04-12
WO2007017468A2 (en) 2007-02-15
JP2009503034A (ja) 2009-01-29
PE20070415A1 (es) 2007-05-29
KR20080040695A (ko) 2008-05-08
RU2008108089A (ru) 2009-09-10
WO2007017468A3 (en) 2007-05-03
MX2008001611A (es) 2008-02-19
CA2617720A1 (en) 2007-02-15

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