AR039691A1 - Formas de dosificacion solidas farmaceuticas - Google Patents
Formas de dosificacion solidas farmaceuticasInfo
- Publication number
- AR039691A1 AR039691A1 ARP030102145A ARP030102145A AR039691A1 AR 039691 A1 AR039691 A1 AR 039691A1 AR P030102145 A ARP030102145 A AR P030102145A AR P030102145 A ARP030102145 A AR P030102145A AR 039691 A1 AR039691 A1 AR 039691A1
- Authority
- AR
- Argentina
- Prior art keywords
- weight
- ethanomidoylamino
- thio
- antioxidant
- ethyl
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P23/00—Anaesthetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pulmonology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Anesthesiology (AREA)
- Pain & Pain Management (AREA)
- Otolaryngology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
Abstract
Se describen composiciones farmacéuticas que comprenden (2S)-2-amino-4-{[2-(etanomidoilamino)etil]tio}butanoico, de fórmula general (1): un agente de relleno farmacéuticamente aceptable y uno o más agentes antioxidantes o quelantes. Reivindicación 6: Una composición farmacéutica de acuerdo con una cualquiera de las reivindicaciones 1 a 5, en la que el ácido (2S)-2-amino-4-{[2-(etanomidoilamino)etil]tio}butanoico comprende de aproximadamente un 0,1 a aproximadamente un 5% en peso, el agente de relleno farmacéuticamente aceptable comprende de aproximadamente un 80 a aproximadamente un 99,5% en peso y el agente antioxidante y quelante, o mezcla de los mismos comprende de aproximadamente un 0,005 a aproximadamente un 5% en peso, con respecto al peso seco. Reivindicación 12: Uso de una composición farmacéutica de acuerdo con cualquiera de las reivindicaciones 1 a 8 en la fabricación de un medicamento para la profilaxis o tratamiento de una afección clínica para la que está indicado un inhibidor de la óxido nítrico sintasa. Reivindicación 13: Uso de acuerdo con la reivindicación 12, en la que la afección clínica se selecciona entre artritis, asma, rinitis, enfermedad pulmonar obstructiva crónica, íleo, migrana, dolor y síndrome del intestino irritable.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0214147.1A GB0214147D0 (en) | 2002-06-19 | 2002-06-19 | Formulations |
Publications (1)
Publication Number | Publication Date |
---|---|
AR039691A1 true AR039691A1 (es) | 2005-03-09 |
Family
ID=9938915
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP030102145A AR039691A1 (es) | 2002-06-19 | 2003-06-17 | Formas de dosificacion solidas farmaceuticas |
Country Status (8)
Country | Link |
---|---|
US (1) | US20050222260A1 (es) |
EP (1) | EP1513511A1 (es) |
JP (1) | JP2005533075A (es) |
AR (1) | AR039691A1 (es) |
AU (1) | AU2003278958A1 (es) |
GB (1) | GB0214147D0 (es) |
TW (1) | TW200404766A (es) |
WO (1) | WO2004000296A1 (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1750675B1 (en) * | 2004-06-02 | 2008-10-29 | Galephar M/F | Stable oral pharmaceutical compositions of buprenorphine and salt thereof |
WO2011052499A1 (ja) * | 2009-10-28 | 2011-05-05 | 第一三共株式会社 | 貯蔵安定性が改善された医薬組成物 |
DE102011051304A1 (de) * | 2011-06-24 | 2012-12-27 | Hennig Arzneimittel Gmbh & Co. Kg | Wirkstoffmatrix |
CN102908323B (zh) * | 2012-10-30 | 2015-03-04 | 天津红日药业股份有限公司 | 一种含有莫西沙星的药物组合物 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NZ289157A (en) * | 1994-06-15 | 1998-03-25 | Wellcome Found | Amidino sulphoxides and sulphones; medicaments for selective inhibition of inducible nitric oxide synthase |
CA2194371A1 (en) * | 1994-07-04 | 1996-01-18 | Thomas Backensfeld | Low-dose steroid tablets containing gallic acid esters as antioxidant agent, process for the manufacture of said tablets, and uses of said tablets |
FR2753098B1 (fr) * | 1996-09-06 | 1998-11-27 | Sod Conseils Rech Applic | Composition pharmaceutique comprenant au moins un inhibiteur de no synthase et au moins un piegeur des formes reactives de l'oxygene |
MY117948A (en) * | 1997-01-13 | 2004-08-30 | Glaxo Group Ltd | Nitride oxide synthase inhibitors. |
GB0031179D0 (en) * | 2000-12-21 | 2001-01-31 | Glaxo Group Ltd | Nitric oxide synthase inhibitors |
-
2002
- 2002-06-19 GB GBGB0214147.1A patent/GB0214147D0/en not_active Ceased
-
2003
- 2003-06-17 TW TW092116417A patent/TW200404766A/zh unknown
- 2003-06-17 AR ARP030102145A patent/AR039691A1/es unknown
- 2003-06-19 JP JP2004514780A patent/JP2005533075A/ja active Pending
- 2003-06-19 AU AU2003278958A patent/AU2003278958A1/en not_active Abandoned
- 2003-06-19 US US10/517,801 patent/US20050222260A1/en not_active Abandoned
- 2003-06-19 EP EP03740281A patent/EP1513511A1/en not_active Withdrawn
- 2003-06-19 WO PCT/EP2003/006465 patent/WO2004000296A1/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
EP1513511A1 (en) | 2005-03-16 |
AU2003278958A1 (en) | 2004-01-06 |
JP2005533075A (ja) | 2005-11-04 |
TW200404766A (en) | 2004-04-01 |
GB0214147D0 (en) | 2002-07-31 |
US20050222260A1 (en) | 2005-10-06 |
WO2004000296A1 (en) | 2003-12-31 |
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