AR005009A1 - Monohidrato del cdch, procedimiento para su produccion , composiciones antibacteriales que lo contienen, uso del monohidrato del cdch para la manufactura de medicamentos. - Google Patents

Monohidrato del cdch, procedimiento para su produccion , composiciones antibacteriales que lo contienen, uso del monohidrato del cdch para la manufactura de medicamentos.

Info

Publication number
AR005009A1
AR005009A1 ARP960105569A ARP960105569A AR005009A1 AR 005009 A1 AR005009 A1 AR 005009A1 AR P960105569 A ARP960105569 A AR P960105569A AR P960105569 A ARP960105569 A AR P960105569A AR 005009 A1 AR005009 A1 AR 005009A1
Authority
AR
Argentina
Prior art keywords
cdch monohydrate
cdch
monohydrate
medicines
procedure
Prior art date
Application number
ARP960105569A
Other languages
English (en)
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7779831&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR005009(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Publication of AR005009A1 publication Critical patent/AR005009A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
ARP960105569A 1995-12-12 1996-12-09 Monohidrato del cdch, procedimiento para su produccion , composiciones antibacteriales que lo contienen, uso del monohidrato del cdch para la manufactura de medicamentos. AR005009A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19546249A DE19546249A1 (de) 1995-12-12 1995-12-12 Neue Kristallmodifikation des 1-Cyclopropyl-7-([S,S]-2,8-diazabicyclo[4,3,0]non-8-yl)-6-fluor-1,4-dihydro-8-methoxy-4-oxo-3-chinolincarbonsäure Hydrochlorid (CDCH), Verfahren zu dessen Herstellung und diese enthaltende pharmazeutische Zubereitungen

Publications (1)

Publication Number Publication Date
AR005009A1 true AR005009A1 (es) 1999-04-07

Family

ID=7779831

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP960105569A AR005009A1 (es) 1995-12-12 1996-12-09 Monohidrato del cdch, procedimiento para su produccion , composiciones antibacteriales que lo contienen, uso del monohidrato del cdch para la manufactura de medicamentos.

Country Status (42)

Country Link
US (1) US5849752A (es)
EP (1) EP0780390B1 (es)
JP (1) JP4104687B2 (es)
KR (1) KR100525146B1 (es)
CN (1) CN1061348C (es)
AR (1) AR005009A1 (es)
AT (1) ATE221531T1 (es)
AU (1) AU708006B2 (es)
BG (1) BG62258B1 (es)
BR (1) BR9605968A (es)
CA (1) CA2192418C (es)
CO (1) CO4480105A1 (es)
CU (1) CU22774A3 (es)
CZ (1) CZ288657B6 (es)
DE (2) DE19546249A1 (es)
DK (1) DK0780390T3 (es)
EE (1) EE03474B1 (es)
ES (1) ES2179910T3 (es)
HR (1) HRP960558B1 (es)
HU (1) HU226521B1 (es)
ID (1) ID22625A (es)
IL (1) IL119795A (es)
IN (1) IN185805B (es)
MA (1) MA24342A1 (es)
MY (1) MY117492A (es)
NL (1) NL300109I1 (es)
NO (1) NO306725B1 (es)
NZ (1) NZ299905A (es)
PL (1) PL184885B1 (es)
PT (1) PT780390E (es)
RO (1) RO119782B1 (es)
RU (1) RU2162468C2 (es)
SA (1) SA96170492B1 (es)
SG (1) SG47201A1 (es)
SI (1) SI0780390T1 (es)
SK (1) SK282805B6 (es)
SV (1) SV1996000109A (es)
TR (1) TR199600970A2 (es)
TW (1) TW411340B (es)
UA (1) UA35638C2 (es)
YU (1) YU49485B (es)
ZA (1) ZA9610405B (es)

Families Citing this family (35)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL134591A0 (en) * 1997-09-25 2001-04-30 Bayer Ag Medicament formulation with a controlled release of an active agent
DE19751948A1 (de) * 1997-11-24 1999-05-27 Bayer Ag Verfahren zur Herstellung von 8-Methoxy-Chinoloncarbonsäuren
US6716830B2 (en) 1998-09-30 2004-04-06 Alcon, Inc. Ophthalmic antibiotic compositions containing moxifloxacin
US6395746B1 (en) 1998-09-30 2002-05-28 Alcon Manufacturing, Ltd. Methods of treating ophthalmic, otic and nasal infections and attendant inflammation
US6509327B1 (en) 1998-09-30 2003-01-21 Alcon Manufacturing, Ltd. Compositions and methods for treating otic, ophthalmic and nasal infections
AU745282B2 (en) * 1998-11-10 2002-03-21 Bayer Intellectual Property Gmbh Pharmaceutical moxifloxacin preparation
DE19854356A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Kristallmodifikation A von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo-/4.3.0/nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE19854357A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Semi-Hydrochlorid von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo/4.3.0/ -nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE19854355A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Kristallmodifikation B von 8-Cyan-1-cyclopropyl-7-(1S, 6S-2,8-diazabicyclo-/4.3.O/nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE19908449A1 (de) * 1999-02-26 2000-08-31 Bayer Ag Kristallmodifikation C von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicylo-[4.3.0]nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chino/incarbonsäure
US20060252789A1 (en) * 2002-10-31 2006-11-09 Sujay Biswas Amorphous moxifloxacin hydrochloride
EP1615645B2 (en) 2003-04-09 2013-08-21 Dr. Reddy's Laboratories Ltd. A crystalline form iii of anhydrous moxifloxacin hydrochloride and a process for the preparation thereof
WO2005012285A1 (en) * 2003-08-05 2005-02-10 Matrix Laboratories Ltd An improved process for the preparation of moxifloxacin hydrochloride
ITMI20032259A1 (it) 2003-11-20 2005-05-21 Chemi Spa Nuovo polimorfo dell'acido 1-ciclopropil-7-(s,s-2,8-diazabciclo-4.3.0-non-8-il)-6-fluoro-1,4-diidro-8-metossi-4-oxo-chinolin carbossilico cloridrato e metodi per la sua preparazione
EP1685130B1 (en) * 2003-11-20 2008-12-10 CHEMI S.p.A. Polymorphs of 1-cyclopropyl-7-([s,s] - 2,8-diazadicyclo [4.3.0] non-8-yl) -6-fluoro-1,4-dihydro-8-methoxy-4-oxo-3-quinoline carboxylic acid hydrochloride and methods for the preparation thereof
US7491725B2 (en) 2004-02-06 2009-02-17 Bristol-Myers Squibb Company Process for preparing 2-aminothiazole-5-aromatic carboxamides as kinase inhibitors
DE102004063347A1 (de) * 2004-12-23 2006-07-13 Stada Arzneimittel Ag Gebrauchsfertige Gemcitabinlösungen und Gemcitabinlösungskonzentrate
WO2007033515A1 (fr) * 2005-09-21 2007-03-29 Shenzhen Tys R & D Co., Ltd. Formulation orale contenant de la moxifloxacine et son procédé de préparation
GB0612422D0 (en) * 2006-06-23 2006-08-02 Generics Uk Ltd Novel hydrate form
CA2655061A1 (en) 2006-06-27 2008-01-03 Sandoz Ag New method for salt preparation
ES2303768B1 (es) * 2006-09-08 2009-06-05 Quimica Sintetica, S.A. Nueva forma cristalina de moxifloxacino clorhidrato.
EP2089388B1 (en) * 2006-11-13 2014-01-29 Cipla Limited Process for the synthesis of moxifloxacin hydrochloride
EP1992626A1 (en) * 2007-05-10 2008-11-19 Sandoz AG Process for the preparation of moxifloxacin hydrochloride
EP2083010A1 (en) * 2008-01-08 2009-07-29 Chemo Ibérica, S.A. Polymorphic Forms of Moxifloxacin hydrochloride and processes for preparation thereof
EP2154137A1 (en) 2008-08-04 2010-02-17 Chemo Ibérica, S.A. Crystalline form of moxifloxacin base
US8314122B2 (en) 2008-10-09 2012-11-20 Abdi Ibrahim Ilac Sanayi Ve Ticaret Anonim Sirketi Using of organic solvents in wet granulation of moxifloxacin
WO2010052726A1 (en) * 2008-11-06 2010-05-14 Hetero Research Foundation Novel polymorph of moxifloxacin hydrochloride
EP2735307A1 (de) 2008-12-08 2014-05-28 Ratiopharm GmbH Kompaktiertes Moxifloxacin
AU2010247141A1 (en) 2009-05-15 2011-12-15 Redx Pharma Plc Redox drug derivatives
WO2011121596A2 (en) * 2010-04-01 2011-10-06 Neuland Laboratories Ltd. Crystal modification of moxifloxacin hydrochloride
BRPI1106900A2 (pt) 2011-12-26 2013-11-05 Ems Sa Composição farmacêutica sólida compreendendo antibótico da familia das quinolonas e processo de sua obtenção
FR2992218B1 (fr) 2012-06-22 2015-01-23 Rivopharm Sa Composition pharmaceutique de chlorhydrate de moxifloxacine et procede de preparation
CN102924449B (zh) * 2012-10-30 2015-08-12 重庆福安药业集团庆余堂制药有限公司 盐酸莫西沙星h晶型及其制备方法和药物组合物
EP2928892B1 (en) 2012-12-04 2018-03-21 Mankind Pharma Ltd. An improved process for the preparation of moxifloxacin hydrochloride
RU2561037C2 (ru) * 2013-02-07 2015-08-20 Открытое акционерное общество "Химико-фармацевтический комбинат "АКРИХИН" (ОАО "АКРИХИН") Антибактериальная фармацевтическая композиция и способ ее получения

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3601567A1 (de) * 1986-01-21 1987-07-23 Bayer Ag 7-(azabicycloalkyl)-chinoloncarbonsaeure- und -naphthyridon-carbonsaeure-derivate
CN1019114B (zh) * 1986-03-31 1992-11-18 三共株式会社 喹啉-3-羟酸衍生物的制备方法
AU609974B2 (en) * 1988-05-18 1991-05-09 Warner-Lambert Company Improved process for the preparation of 5-amino-7- (substituted amino)-quinoline-3-carboxylic acids
DE3910663A1 (de) * 1989-04-03 1990-10-04 Bayer Ag 5-alkylchinoloncarbonsaeuren
TW209865B (es) 1992-01-10 1993-07-21 Bayer Ag
CA2128601C (en) * 1992-01-31 2003-07-15 Hiroyuki Nagano Quinolone carboxylic acid derivatives in crystalline hydrate form
DE4234078A1 (de) 1992-10-09 1994-04-14 Bayer Ag Chinoloncarbonsäuren
CA2112165C (en) * 1992-12-25 2003-04-08 Makoto Takemura Bicyclic amine derivatives
ZA946853B (en) * 1993-09-10 1995-04-24 Daiichi Seiyaku Co Crystals of antimicrobial compound.
DK0676199T3 (da) * 1994-04-07 1999-02-08 Pfizer Anvendelse af trovafloxacin eller derivater deraf til fremstilling af et medikament til behandling af H. pylori-infektione

Also Published As

Publication number Publication date
KR100525146B1 (ko) 2006-01-27
NZ299905A (en) 1998-09-24
JP4104687B2 (ja) 2008-06-18
ES2179910T3 (es) 2003-02-01
JPH09169757A (ja) 1997-06-30
CN1061348C (zh) 2001-01-31
YU65096A (sh) 1998-12-23
TR199600970A2 (tr) 1997-06-21
IN185805B (es) 2001-05-05
SK159196A3 (en) 1997-10-08
ID22625A (id) 1999-12-02
DK0780390T3 (da) 2002-11-11
RU2162468C2 (ru) 2001-01-27
EP0780390A1 (de) 1997-06-25
CA2192418A1 (en) 1997-06-13
EE03474B1 (et) 2001-08-15
CZ288657B6 (cs) 2001-08-15
NO965298D0 (no) 1996-12-11
BG62258B1 (bg) 1999-06-30
CA2192418C (en) 2001-06-12
AU708006B2 (en) 1999-07-29
ATE221531T1 (de) 2002-08-15
IL119795A0 (en) 1997-03-18
EE9600201A (et) 1997-06-16
BR9605968A (pt) 1998-08-18
NO965298L (no) 1997-06-13
PT780390E (pt) 2002-11-29
KR970042550A (ko) 1997-07-24
EP0780390B1 (de) 2002-07-31
SA96170492B1 (ar) 2006-05-23
ZA9610405B (en) 1997-06-23
DE59609501D1 (de) 2002-09-05
MA24342A1 (fr) 1998-07-01
CZ364696A3 (en) 1997-07-16
MY117492A (en) 2004-07-31
IL119795A (en) 1998-12-27
NL300109I1 (nl) 2003-02-03
HRP960558B1 (en) 2002-04-30
RO119782B1 (ro) 2005-03-30
CN1160052A (zh) 1997-09-24
SG47201A1 (en) 1998-03-20
HU9603428D0 (en) 1997-01-28
HUP9603428A2 (en) 1997-08-28
NO306725B1 (no) 1999-12-13
HUP9603428A3 (en) 1997-10-28
HU226521B1 (en) 2009-03-30
YU49485B (sh) 2006-08-17
SV1996000109A (es) 1997-10-23
AU7421696A (en) 1997-06-19
PL184885B1 (pl) 2003-01-31
SK282805B6 (sk) 2002-12-03
DE19546249A1 (de) 1997-06-19
CO4480105A1 (es) 1997-07-09
HRP960558A2 (en) 1998-02-28
SI0780390T1 (en) 2002-10-31
PL317415A1 (en) 1997-06-23
US5849752A (en) 1998-12-15
MX9606325A (es) 1997-10-31
TW411340B (en) 2000-11-11
BG101043A (en) 1998-04-30
CU22774A3 (es) 2002-07-24
UA35638C2 (uk) 2001-04-16

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