DK226983D0 - Fremgangsmade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre - Google Patents

Fremgangsmade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre

Info

Publication number
DK226983D0
DK226983D0 DK2269/83A DK226983A DK226983D0 DK 226983 D0 DK226983 D0 DK 226983D0 DK 2269/83 A DK2269/83 A DK 2269/83A DK 226983 A DK226983 A DK 226983A DK 226983 D0 DK226983 D0 DK 226983D0
Authority
DK
Denmark
Prior art keywords
methylammonium
derivatives
preparing
dioxopenicillanic acid
dioxopenicillanic
Prior art date
Application number
DK2269/83A
Other languages
English (en)
Other versions
DK226983A (da
Inventor
Robert Fischer Myers
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK226983D0 publication Critical patent/DK226983D0/da
Publication of DK226983A publication Critical patent/DK226983A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK226983A 1982-05-24 1983-05-20 Fremgangsmaade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre DK226983A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/381,104 US4428935A (en) 1982-05-24 1982-05-24 Penicillanic acid dioxide prodrug

Publications (2)

Publication Number Publication Date
DK226983D0 true DK226983D0 (da) 1983-05-20
DK226983A DK226983A (da) 1983-11-25

Family

ID=23503664

Family Applications (1)

Application Number Title Priority Date Filing Date
DK226983A DK226983A (da) 1982-05-24 1983-05-20 Fremgangsmaade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre

Country Status (7)

Country Link
US (1) US4428935A (da)
EP (1) EP0095341B1 (da)
JP (1) JPS58216191A (da)
DE (1) DE3362266D1 (da)
DK (1) DK226983A (da)
GR (1) GR79260B (da)
IE (1) IE55577B1 (da)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4946959A (en) * 1984-11-30 1990-08-07 The Dow Chemical Company Method of preparing 5-alkyl-1-(2-pyridinyl)-1H-1,2,4-triazol-3-ols
US4681943A (en) * 1984-11-30 1987-07-21 The Dow Chemical Company 1-acyl-1-(2-pyridinyl)semicarbazides
WO1991016326A1 (en) * 1990-04-13 1991-10-31 Pfizer Inc. Process for sultamicillin intermediate
US7189351B2 (en) * 2001-10-25 2007-03-13 Spherix Incorporated D-tagatose as an anti-biofilm agent
PA8579701A1 (es) * 2002-08-23 2005-05-24 Pfizer Prod Inc Profarmaco inhibidor de beta-lactamasa
WO2004108733A1 (en) * 2003-06-05 2004-12-16 Pfizer Products Inc. Beta-lactamase inhibitor prodrug
JP2007534771A (ja) * 2004-04-27 2007-11-29 メディシノバ,インコーポレーテッド 炎症性疾患の治療におけるフェノキシアルキルカルボン酸誘導体
ES2547258T3 (es) 2006-12-10 2015-10-02 Chongxi Yu Sistemas de administración transdérmica de antibióticos beta-lactama
CN105566213B (zh) * 2009-06-10 2019-11-12 上海泰飞尔生化技术有限公司 具有高穿透性的抗微生物剂和抗微生物剂相关化合物的前药组合物
US9969751B2 (en) 2009-06-10 2018-05-15 Techfields Pharma Co., Ltd. High penetration prodrug compositions of antimicrobials and antimicrobial-related compounds
HRP20171415T4 (hr) 2009-06-25 2023-03-03 Alkermes Pharma Ireland Limited Heterociklični spojevi za liječenje neuroloških i psiholoških poremećaja
WO2010151711A1 (en) 2009-06-25 2010-12-29 Alkermes, Inc. Prodrugs of nh-acidic compounds
WO2011163594A2 (en) 2010-06-24 2011-12-29 Alkermes, Inc. Prodrugs of nh-acidic compounds: ester, carbonate, carbamate and phosphonate derivatives
CN103561746B (zh) 2011-03-18 2018-05-29 奥克梅斯制药爱尔兰有限公司 包含脱水山梨糖醇酯的药物组合物
PL2736510T3 (pl) * 2011-07-28 2017-07-31 Kempharm, Inc. Proleki metylofenidatu, procesy ich wytwarzania i stosowania
NZ722096A (en) 2011-12-15 2016-11-25 Alkermes Pharma Ireland Ltd Prodrugs of secondary amine compounds
EP2827868B8 (en) 2012-03-19 2019-12-18 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising fatty acid esters
CA2867137C (en) 2012-03-19 2020-12-08 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising aripiprazole prodrugs and benzyl alcohol
CA2867123C (en) 2012-03-19 2021-02-16 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising water-insoluble antipsychotic agents and glycerol esters
CA2885196C (en) 2012-09-19 2021-06-22 Alkermes Pharma Ireland Limited Pharmaceutical compositions having improved storage stability
US9556156B2 (en) * 2012-10-05 2017-01-31 Sphaera Pharma Pte Ltd. Compounds, their synthesis and their uses
CN110368360A (zh) 2014-03-20 2019-10-25 奥克梅斯制药爱尔兰有限公司 具有增加的注射速度的阿立哌唑制剂
CN112423754A (zh) 2018-03-05 2021-02-26 奥克梅斯制药爱尔兰有限公司 阿立哌唑的给药策略
CA3175830A1 (en) * 2019-04-17 2020-10-22 Sundeep Dugar Prodrugs of monomethyl fumarate

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1255034A (en) * 1968-09-06 1971-11-24 Beecham Group Ltd Penicillin esters
NL7401782A (da) * 1973-02-14 1974-08-16
US4234579A (en) 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
JPS6056160B2 (ja) 1977-06-07 1985-12-09 フアイザ−・インコ−ポレ−テツド β−ラクタマ−ゼ阻害剤としてのペニシラン酸1,1−ジオキシド
US4244951A (en) 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
US4376767A (en) * 1981-01-02 1983-03-15 Merck & Co., Inc. Pyridylmethyl esters of selected bio-affecting carboxylic acids
US4323499A (en) 1981-01-05 1982-04-06 Pfizer Inc. 6-(2-Aryl-2-(1,1-dioxopenicillanoyloxy-methoxycarbonyl)acetamido penicillanic acids

Also Published As

Publication number Publication date
JPS58216191A (ja) 1983-12-15
EP0095341A1 (en) 1983-11-30
DK226983A (da) 1983-11-25
IE55577B1 (en) 1990-11-07
GR79260B (da) 1984-10-22
US4428935A (en) 1984-01-31
DE3362266D1 (de) 1986-04-03
EP0095341B1 (en) 1986-02-26
IE831203L (en) 1983-11-24

Similar Documents

Publication Publication Date Title
DK226983A (da) Fremgangsmaade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre
DK336783D0 (da) Fremgangsmade til fremstilling af methylendiphosphonsyrederivater
DK144783D0 (da) Fremgangsmade til fremstilling af cycloalka(c)pyrrol-carboxylsyrederivater
DK361281A (da) Fremgangsmaade til fremstilling af 2,5-diketo-d-gluconsyre
DK90494A (da) Fremgangsmåde til fremstilling af 2,3,4,5,-tetrafluorbenzoesyre
DK166087C (da) Fremgangsmaade til fremstilling af oe(3-amino-3-carboxy)-propyl-1aaphosphinsyrederivater
DK357782A (da) Fremgangsmaade til fremstilling af tetrahydrofurancarboxylsyrederivater
DK103583A (da) Fremgangsmaade til fremstilling af 2-keto-l-gulonsyre
DK533881A (da) Fremgangsmaade til fremstilling af 3,4-bis-substituerede 1,2,5-oxidazol-2-oxider eller farmekologisk acceptable syreadditionsforbindelser
DK436685A (da) Fremgangsmaade til fremstilling af 2,4-dichlor-5-fluor-benzoesyre
DK24083D0 (da) Fremgangsmade til fremstilling af 0,0'-dithiodibenzoesyrer
DK433987D0 (da) Fremgangsmaade til fremstilling af 1,12-dodecandisyre ii
DK162997C (da) Fremgangsmaade til fremstilling af 5,6,7,8-tetrahydrofolinsyre
DK154085C (da) Fremgangsmaade til fremstilling af 1,1-dioxopenicillansyrederivater
DK87382A (da) Fremgangsmaade til fremstilling af 1,4,5,6,7,8-hexahydro-2-alkyl-4-aryl-5-oxo-1,7-naphthyridin-3-carboxylsyreestere
DK454183A (da) Fremgangsmaade til fremstilling af 15-cycloaliphatiske derivater af 13,14-didehydro-carboprostancycliner
DK228583D0 (da) Fremgangsmade til fremstilling af 5-oxo-2-pyrrolidinpropansyrederivater
DK149962C (da) Fremgangsmaade til fremstilling af 2,5-diketogluconsyre
DK154969C (da) Fremgangsmaade til fremstilling af nicotinylesteren af 6-aminonicotinsyre
DK162768C (da) Fremgangsmaade til fremstilling af oxazolinoazetidinylhydroxymethylbutensyrederivater
DK477682A (da) Fremgangsmaade til fremstilling af aminocyklopentanalkensyrer
DK496682A (da) Fremgangsmaade til fremstilling af beta-hydroxy-beta-methylglutarsyre
DK310583A (da) Fremgangsmaade til fremstilling af 7-amino-1-dethia-1-oxa-3-hydroxymethyl-cephem-4-carboxylsyrer
DK164680A (da) Fremgangsmaade til fremstilling af 2,3-dihydroxybenzoesyre
DK160819C (da) Fremgangsmaade til fremstilling af 3,5-dichlor-2-pyridon

Legal Events

Date Code Title Description
AHB Application shelved due to non-payment