DK226983D0 - Fremgangsmade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre - Google Patents
Fremgangsmade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyreInfo
- Publication number
- DK226983D0 DK226983D0 DK2269/83A DK226983A DK226983D0 DK 226983 D0 DK226983 D0 DK 226983D0 DK 2269/83 A DK2269/83 A DK 2269/83A DK 226983 A DK226983 A DK 226983A DK 226983 D0 DK226983 D0 DK 226983D0
- Authority
- DK
- Denmark
- Prior art keywords
- methylammonium
- derivatives
- preparing
- dioxopenicillanic acid
- dioxopenicillanic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US06/381,104 US4428935A (en) | 1982-05-24 | 1982-05-24 | Penicillanic acid dioxide prodrug |
Publications (2)
Publication Number | Publication Date |
---|---|
DK226983D0 true DK226983D0 (da) | 1983-05-20 |
DK226983A DK226983A (da) | 1983-11-25 |
Family
ID=23503664
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK226983A DK226983A (da) | 1982-05-24 | 1983-05-20 | Fremgangsmaade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre |
Country Status (7)
Country | Link |
---|---|
US (1) | US4428935A (da) |
EP (1) | EP0095341B1 (da) |
JP (1) | JPS58216191A (da) |
DE (1) | DE3362266D1 (da) |
DK (1) | DK226983A (da) |
GR (1) | GR79260B (da) |
IE (1) | IE55577B1 (da) |
Families Citing this family (24)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4946959A (en) * | 1984-11-30 | 1990-08-07 | The Dow Chemical Company | Method of preparing 5-alkyl-1-(2-pyridinyl)-1H-1,2,4-triazol-3-ols |
US4681943A (en) * | 1984-11-30 | 1987-07-21 | The Dow Chemical Company | 1-acyl-1-(2-pyridinyl)semicarbazides |
WO1991016326A1 (en) * | 1990-04-13 | 1991-10-31 | Pfizer Inc. | Process for sultamicillin intermediate |
US7189351B2 (en) * | 2001-10-25 | 2007-03-13 | Spherix Incorporated | D-tagatose as an anti-biofilm agent |
PA8579701A1 (es) * | 2002-08-23 | 2005-05-24 | Pfizer Prod Inc | Profarmaco inhibidor de beta-lactamasa |
WO2004108733A1 (en) * | 2003-06-05 | 2004-12-16 | Pfizer Products Inc. | Beta-lactamase inhibitor prodrug |
JP2007534771A (ja) * | 2004-04-27 | 2007-11-29 | メディシノバ,インコーポレーテッド | 炎症性疾患の治療におけるフェノキシアルキルカルボン酸誘導体 |
ES2547258T3 (es) | 2006-12-10 | 2015-10-02 | Chongxi Yu | Sistemas de administración transdérmica de antibióticos beta-lactama |
CN105566213B (zh) * | 2009-06-10 | 2019-11-12 | 上海泰飞尔生化技术有限公司 | 具有高穿透性的抗微生物剂和抗微生物剂相关化合物的前药组合物 |
US9969751B2 (en) | 2009-06-10 | 2018-05-15 | Techfields Pharma Co., Ltd. | High penetration prodrug compositions of antimicrobials and antimicrobial-related compounds |
HRP20171415T4 (hr) | 2009-06-25 | 2023-03-03 | Alkermes Pharma Ireland Limited | Heterociklični spojevi za liječenje neuroloških i psiholoških poremećaja |
WO2010151711A1 (en) | 2009-06-25 | 2010-12-29 | Alkermes, Inc. | Prodrugs of nh-acidic compounds |
WO2011163594A2 (en) | 2010-06-24 | 2011-12-29 | Alkermes, Inc. | Prodrugs of nh-acidic compounds: ester, carbonate, carbamate and phosphonate derivatives |
CN103561746B (zh) | 2011-03-18 | 2018-05-29 | 奥克梅斯制药爱尔兰有限公司 | 包含脱水山梨糖醇酯的药物组合物 |
PL2736510T3 (pl) * | 2011-07-28 | 2017-07-31 | Kempharm, Inc. | Proleki metylofenidatu, procesy ich wytwarzania i stosowania |
NZ722096A (en) | 2011-12-15 | 2016-11-25 | Alkermes Pharma Ireland Ltd | Prodrugs of secondary amine compounds |
EP2827868B8 (en) | 2012-03-19 | 2019-12-18 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising fatty acid esters |
CA2867137C (en) | 2012-03-19 | 2020-12-08 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising aripiprazole prodrugs and benzyl alcohol |
CA2867123C (en) | 2012-03-19 | 2021-02-16 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising water-insoluble antipsychotic agents and glycerol esters |
CA2885196C (en) | 2012-09-19 | 2021-06-22 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions having improved storage stability |
US9556156B2 (en) * | 2012-10-05 | 2017-01-31 | Sphaera Pharma Pte Ltd. | Compounds, their synthesis and their uses |
CN110368360A (zh) | 2014-03-20 | 2019-10-25 | 奥克梅斯制药爱尔兰有限公司 | 具有增加的注射速度的阿立哌唑制剂 |
CN112423754A (zh) | 2018-03-05 | 2021-02-26 | 奥克梅斯制药爱尔兰有限公司 | 阿立哌唑的给药策略 |
CA3175830A1 (en) * | 2019-04-17 | 2020-10-22 | Sundeep Dugar | Prodrugs of monomethyl fumarate |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1255034A (en) * | 1968-09-06 | 1971-11-24 | Beecham Group Ltd | Penicillin esters |
NL7401782A (da) * | 1973-02-14 | 1974-08-16 | ||
US4234579A (en) | 1977-06-07 | 1980-11-18 | Pfizer Inc. | Penicillanic acid 1,1-dioxides as β-lactamase inhibitors |
JPS6056160B2 (ja) | 1977-06-07 | 1985-12-09 | フアイザ−・インコ−ポレ−テツド | β−ラクタマ−ゼ阻害剤としてのペニシラン酸1,1−ジオキシド |
US4244951A (en) | 1979-05-16 | 1981-01-13 | Pfizer Inc. | Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide |
US4376767A (en) * | 1981-01-02 | 1983-03-15 | Merck & Co., Inc. | Pyridylmethyl esters of selected bio-affecting carboxylic acids |
US4323499A (en) | 1981-01-05 | 1982-04-06 | Pfizer Inc. | 6-(2-Aryl-2-(1,1-dioxopenicillanoyloxy-methoxycarbonyl)acetamido penicillanic acids |
-
1982
- 1982-05-24 US US06/381,104 patent/US4428935A/en not_active Expired - Lifetime
-
1983
- 1983-05-20 DK DK226983A patent/DK226983A/da not_active Application Discontinuation
- 1983-05-20 DE DE8383302891T patent/DE3362266D1/de not_active Expired
- 1983-05-20 EP EP83302891A patent/EP0095341B1/en not_active Expired
- 1983-05-23 GR GR71431A patent/GR79260B/el unknown
- 1983-05-23 IE IE1203/83A patent/IE55577B1/en unknown
- 1983-05-24 JP JP58091409A patent/JPS58216191A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
JPS58216191A (ja) | 1983-12-15 |
EP0095341A1 (en) | 1983-11-30 |
DK226983A (da) | 1983-11-25 |
IE55577B1 (en) | 1990-11-07 |
GR79260B (da) | 1984-10-22 |
US4428935A (en) | 1984-01-31 |
DE3362266D1 (de) | 1986-04-03 |
EP0095341B1 (en) | 1986-02-26 |
IE831203L (en) | 1983-11-24 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
AHB | Application shelved due to non-payment |