BG21230A3 - Метод за получаване на n/ хетероарилметил/ д7- дезокси - норморфини и- норкодеини - Google Patents

Метод за получаване на n/ хетероарилметил/ д7- дезокси - норморфини и- норкодеини

Info

Publication number: BG21230A3
Authority: BG; Bulgaria
Prior art keywords: normorphines; norcodeines; deoxys; heteroarylmethyl; obtaining
Prior art date: 1972-09-14

Application number

BG025619A

Other languages

Bulgarian (bg)

English (en)

Inventor

Gerhard Walther

Adolf Merz

Herbert Merz

Adolf Langbein

Klaus Stockhaus

Original Assignee

C.H.Boehringer Sohn

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1972-09-14

Filing date

1973-09-12

Publication date

1976-03-20

1973-09-12 Application filed by C.H.Boehringer Sohn filed Critical C.H.Boehringer Sohn

1976-03-20 Publication of BG21230A3 publication Critical patent/BG21230A3/xx

Links

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D489/00—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Life Sciences & Earth Sciences (AREA)
Emergency Medicine (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Networks Using Active Elements (AREA)

BG025619A 1972-09-14 1973-09-12 Метод за получаване на n/ хетероарилметил/ д7- дезокси - норморфини и- норкодеини BG21230A3 (bg)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE2245141A DE2245141A1 (de)	1972-09-14	1972-09-14	Neue n-(heteroarylmethyl)-desoxynormorphine und -norcodeine, deren saeureadditionssalze, verfahren zu deren herstellung sowie deren verwendung als arzneimittel

Publications (1)

Publication Number	Publication Date
BG21230A3 true BG21230A3 (bg)	1976-03-20

Family

ID=5856355

Family Applications (8)

Application Number	Title	Priority Date	Filing Date
BG25617A BG21228A3 (ja)	1972-09-14	1973-09-12
BG025619A BG21230A3 (bg)	1972-09-14	1973-09-12	Метод за получаване на n/ хетероарилметил/ д7- дезокси - норморфини и- норкодеини
BG24524A BG21412A3 (ja)	1972-09-14	1973-09-12
BG025613A BG21224A3 (bg)	1972-09-14	1973-09-12	Метод за получаване на n/ хетероарил метил- / -д7 дезокси норморфини м норкодеини
BG025614A BG21225A3 (bg)	1972-09-14	1973-09-12	Метод за получаване на n / хетероарил метил/-д7- дезокси- норморфини и наркодеини
BG025616A BG21227A3 (bg)	1972-09-14	1973-09-12	Метод за получаване на n/ хетепоарилметил/ д7- дезокси- норморфини и норкодеини
BG025618A BG21229A3 (bg)	1972-09-14	1973-09-12	Метод за получаване на n/ хетероарилметил/ д7 дезокси- норморфини- норкодеини
BG025615A BG21226A3 (bg)	1972-09-14	1974-01-28	Метод за получаване на n/хетероарилметил/ д7 -де- зокси- нормофини и ниркодеини

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
BG25617A BG21228A3 (ja)	1972-09-14	1973-09-12

Family Applications After (6)

Application Number	Title	Priority Date	Filing Date
BG24524A BG21412A3 (ja)	1972-09-14	1973-09-12
BG025613A BG21224A3 (bg)	1972-09-14	1973-09-12	Метод за получаване на n/ хетероарил метил- / -д7 дезокси норморфини м норкодеини
BG025614A BG21225A3 (bg)	1972-09-14	1973-09-12	Метод за получаване на n / хетероарил метил/-д7- дезокси- норморфини и наркодеини
BG025616A BG21227A3 (bg)	1972-09-14	1973-09-12	Метод за получаване на n/ хетепоарилметил/ д7- дезокси- норморфини и норкодеини
BG025618A BG21229A3 (bg)	1972-09-14	1973-09-12	Метод за получаване на n/ хетероарилметил/ д7 дезокси- норморфини- норкодеини
BG025615A BG21226A3 (bg)	1972-09-14	1974-01-28	Метод за получаване на n/хетероарилметил/ д7 -де- зокси- нормофини и ниркодеини

Country Status (24)

Country	Link
US (1)	US3928359A (ja)
JP (1)	JPS4966700A (ja)
AT (1)	AT326281B (ja)
BE (1)	BE804836A (ja)
BG (8)	BG21228A3 (ja)
CH (7)	CH605958A5 (ja)
CS (8)	CS168678B2 (ja)
DD (1)	DD109384A5 (ja)
DE (1)	DE2245141A1 (ja)
ES (8)	ES418563A1 (ja)
FI (1)	FI55512C (ja)
FR (1)	FR2199982B1 (ja)
GB (1)	GB1449222A (ja)
HU (1)	HU166367B (ja)
IE (1)	IE38320B1 (ja)
IL (1)	IL43216A (ja)
NL (1)	NL7312621A (ja)
NO (1)	NO139482C (ja)
PL (8)	PL91809B1 (ja)
RO (2)	RO63003A (ja)
SE (1)	SE413510B (ja)
SU (8)	SU498911A3 (ja)
YU (2)	YU243973A (ja)
ZA (1)	ZA737289B (ja)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4241065A (en) *	1979-07-02	1980-12-23	E. I. Du Pont De Nemours And Company	Fluoro analogs of hydrocodone and oxycodone useful as analgesics, narcotic antagonists or both
US4236008A (en) *	1978-09-19	1980-11-25	E. I. Du Pont De Nemours And Company	Fluorination of precursors for fluorine analogs of hydrocodone and oxycodone
WO1999038869A1 (en)	1998-01-29	1999-08-05	Monash University	Therapeutic compounds

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE2107989A1 (de) *	1971-02-19	1972-09-07	Boehringer Sohn Ingelheim	N-(Furyl-methy])-morphinane, deren Säureadditionssalze sowie Verfahren zu deren Herstellung

1972
- 1972-09-14 DE DE2245141A patent/DE2245141A1/de active Pending
1973
- 1973-09-03 AT AT761673A patent/AT326281B/de not_active IP Right Cessation
- 1973-09-07 ES ES418563A patent/ES418563A1/es not_active Expired
- 1973-09-11 CH CH207277A patent/CH605958A5/xx not_active IP Right Cessation
- 1973-09-11 CH CH198077A patent/CH589088A5/xx not_active IP Right Cessation
- 1973-09-11 CH CH207177A patent/CH589090A5/xx not_active IP Right Cessation
- 1973-09-11 CH CH207077A patent/CH591490A5/xx not_active IP Right Cessation
- 1973-09-11 CH CH198177A patent/CH589089A5/xx not_active IP Right Cessation
- 1973-09-11 CH CH1298673A patent/CH590287A5/xx not_active IP Right Cessation
- 1973-09-11 CH CH207377A patent/CH591491A5/xx not_active IP Right Cessation
- 1973-09-11 US US396171A patent/US3928359A/en not_active Expired - Lifetime
- 1973-09-12 HU HUBO1463A patent/HU166367B/hu unknown
- 1973-09-12 CS CS286*[A patent/CS168678B2/cs unknown
- 1973-09-12 CS CS285*[A patent/CS168677B2/cs unknown
- 1973-09-12 BG BG25617A patent/BG21228A3/xx unknown
- 1973-09-12 DD DD173479A patent/DD109384A5/xx unknown
- 1973-09-12 CS CS284*[A patent/CS168676B2/cs unknown
- 1973-09-12 BG BG025619A patent/BG21230A3/xx unknown
- 1973-09-12 IE IE1630/73A patent/IE38320B1/xx unknown
- 1973-09-12 BG BG24524A patent/BG21412A3/xx unknown
- 1973-09-12 BG BG025613A patent/BG21224A3/xx unknown
- 1973-09-12 CS CS288*[A patent/CS168680B2/cs unknown
- 1973-09-12 CS CS282*[A patent/CS168674B2/cs unknown
- 1973-09-12 BG BG025614A patent/BG21225A3/xx unknown
- 1973-09-12 CS CS283*[A patent/CS168675B2/cs unknown
- 1973-09-12 BG BG025616A patent/BG21227A3/xx unknown
- 1973-09-12 SU SU1962620A patent/SU498911A3/ru active
- 1973-09-12 CS CS287*[A patent/CS168679B2/cs unknown
- 1973-09-12 CS CS6322A patent/CS168673B2/cs unknown
- 1973-09-12 BG BG025618A patent/BG21229A3/xx unknown
- 1973-09-13 PL PL1973174974A patent/PL91809B1/pl unknown
- 1973-09-13 ZA ZA00737289A patent/ZA737289B/xx unknown
- 1973-09-13 PL PL1973174971A patent/PL91829B1/pl unknown
- 1973-09-13 JP JP48103716A patent/JPS4966700A/ja active Pending
- 1973-09-13 NL NL7312621A patent/NL7312621A/xx not_active Application Discontinuation
- 1973-09-13 PL PL1973174972A patent/PL91807B1/pl unknown
- 1973-09-13 GB GB4314673A patent/GB1449222A/en not_active Expired
- 1973-09-13 RO RO7300076068A patent/RO63003A/ro unknown
- 1973-09-13 PL PL1973174973A patent/PL91808B1/pl unknown
- 1973-09-13 PL PL1973174968A patent/PL90720B1/pl unknown
- 1973-09-13 PL PL1973174969A patent/PL91837B1/pl unknown
- 1973-09-13 NO NO3588/73A patent/NO139482C/no unknown
- 1973-09-13 PL PL1973174970A patent/PL91836B1/pl unknown
- 1973-09-13 YU YU02439/73A patent/YU243973A/xx unknown
- 1973-09-13 PL PL1973165187A patent/PL87721B1/pl unknown
- 1973-09-13 IL IL43216A patent/IL43216A/en unknown
- 1973-09-13 RO RO7382817A patent/RO70193A/ro unknown
- 1973-09-13 BE BE135636A patent/BE804836A/xx unknown
- 1973-09-13 FI FI2853/73A patent/FI55512C/fi active
- 1973-09-14 SE SE7312583A patent/SE413510B/xx unknown
- 1973-09-14 FR FR7333092A patent/FR2199982B1/fr not_active Expired
1974
- 1974-01-28 BG BG025615A patent/BG21226A3/bg unknown
- 1974-09-19 ES ES430202A patent/ES430202A1/es not_active Expired
- 1974-09-19 ES ES430199A patent/ES430199A1/es not_active Expired
- 1974-09-19 ES ES430200A patent/ES430200A1/es not_active Expired
- 1974-09-19 ES ES430201A patent/ES430201A1/es not_active Expired
- 1974-09-19 ES ES430198A patent/ES430198A1/es not_active Expired
- 1974-09-19 ES ES430203A patent/ES430203A1/es not_active Expired
- 1974-09-19 ES ES430197A patent/ES430197A1/es not_active Expired
- 1974-09-30 SU SU2063983A patent/SU509239A3/ru active
- 1974-09-30 SU SU2063984A patent/SU520049A3/ru active
- 1974-09-30 SU SU2063380A patent/SU503524A3/ru active
- 1974-09-30 SU SU2063987A patent/SU506299A3/ru active
- 1974-09-30 SU SU2063985A patent/SU503523A3/ru active
- 1974-09-30 SU SU2063986A patent/SU505366A3/ru active
- 1974-09-30 SU SU2063982A patent/SU528878A3/ru active
1979
- 1979-10-19 YU YU02548/79A patent/YU254879A/xx unknown

Also Published As

Publication number	Publication date
BG21229A3 (bg)	1976-03-20
SU528878A3 (ru)	1976-09-15
CS168678B2 (ja)	1976-06-29
BG21412A3 (ja)	1976-05-20
HU166367B (ja)	1975-03-28
CS168673B2 (ja)	1976-06-29
CH589088A5 (ja)	1977-06-30
SU503523A3 (ru)	1976-02-15
SU506299A3 (ru)	1976-03-05
SU520049A3 (ru)	1976-06-30
BG21225A3 (bg)	1976-03-20
FI55512C (fi)	1979-08-10
ES430203A1 (es)	1976-10-16
RO63003A (fr)	1978-05-15
PL87721B1 (ja)	1976-07-31
NO139482B (no)	1978-12-11
SE413510B (sv)	1980-06-02
CH589089A5 (ja)	1977-06-30
AT326281B (de)	1975-12-10
CH605958A5 (ja)	1978-10-13
CS168674B2 (ja)	1976-06-29
PL91837B1 (ja)	1977-03-31
PL91829B1 (ja)	1977-03-31
NO139482C (no)	1979-03-21
SU498911A3 (ru)	1976-01-05
BG21224A3 (bg)	1976-03-20
BE804836A (fr)	1974-03-13
GB1449222A (en)	1976-09-15
ATA761673A (de)	1975-02-15
ES430198A1 (es)	1976-10-16
ES430197A1 (es)	1976-10-16
BG21228A3 (ja)	1976-03-20
PL91809B1 (ja)	1977-03-31
PL90720B1 (ja)	1977-01-31
CS168680B2 (ja)	1976-06-29
ES430202A1 (es)	1976-10-16
ES430199A1 (es)	1976-10-16
PL91808B1 (ja)	1977-03-31
CS168675B2 (ja)	1976-06-29
JPS4966700A (ja)	1974-06-27
CH590287A5 (ja)	1977-07-29
PL91836B1 (ja)	1977-03-31
ES430201A1 (es)	1976-10-16
YU254879A (en)	1983-01-21
CS168679B2 (ja)	1976-06-29
ES430200A1 (es)	1976-10-16
FR2199982B1 (ja)	1977-01-28
SU503524A3 (ru)	1976-02-15
ZA737289B (en)	1975-05-28
CH591491A5 (ja)	1977-09-30
SU505366A3 (ru)	1976-02-28
IL43216A0 (en)	1973-11-28
CS168677B2 (ja)	1976-06-29
ES418563A1 (es)	1976-05-01
YU243973A (en)	1982-05-31
PL91807B1 (ja)	1977-03-31
RO70193A (ro)	1981-04-30
FI55512B (fi)	1979-04-30
DD109384A5 (ja)	1974-11-05
IE38320B1 (en)	1978-02-15
SU509239A3 (ru)	1976-03-30
US3928359A (en)	1975-12-23
DE2245141A1 (de)	1974-03-21
IL43216A (en)	1976-07-30
CS168676B2 (ja)	1976-06-29
BG21226A3 (bg)	1976-03-20
IE38320L (en)	1974-03-14
AU6030173A (en)	1975-03-13
NL7312621A (ja)	1974-03-18
BG21227A3 (bg)	1976-03-20
FR2199982A1 (ja)	1974-04-19
CH589090A5 (ja)	1977-06-30
CH591490A5 (ja)	1977-09-30

Publication	Publication Date	Title
BG20352A3 (bg)	1975-11-05	Метод за получаване на пиридил-фенил оксиалкани
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BG20816A3 (bg)	1975-12-20	Метод за получаване на дезацетоксицефалоспорини
BG20562A3 (bg)	1975-12-05	Метод за получаване на халогенацетанилиди
BG22826A3 (bg)	1977-04-20	Метод за получаване на оксазоли
BG21230A3 (bg)	1976-03-20	Метод за получаване на n/ хетероарилметил/ д7- дезокси - норморфини и- норкодеини
BG22828A3 (bg)	1977-04-20	Метод за получаване на 2-амино-4-н пирини
BG20778A3 (bg)	1975-12-20	Метод за получаване на 2-алкокси -5- алкилсулфонил - бензоени киселини
BG22808A3 (bg)	1977-04-20	Метод за получаване на базични естери
SU490283A3 (ru)	1975-10-30	Способ получени дифенилметоксиэтиламинов
BG22819A3 (bg)	1977-04-20	Метод за получаване на 3--амино-пиразолони-(5)
BG21223A3 (bg)	1976-03-20	Метод за получаване на м-диоксан-5-метиламини
BG20558A3 (bg)	1975-12-05	Метод за получаване на сирил-пиридини
BG21607A3 (bg)	1976-07-20	Метод за получаване на псевдотризахариди
BG22382A3 (bg)	1977-02-20	Метод за получаване на 2-амино-бензиламини
BG21197A3 (bg)	1976-03-20	Метод за получаване на нови биденилови деривати
BG23007A3 (bg)	1977-05-20	Метод за получаване на циклобутанови производни
SU459193A1 (ru)	1975-02-05	Способ корчевки пней