AR241158A2 - Un procedimiento para la preparacion de compuestos de beta-lactamas y sus sales - Google Patents
Un procedimiento para la preparacion de compuestos de beta-lactamas y sus salesInfo
- Publication number
- AR241158A2 AR241158A2 AR29381583A AR29381583A AR241158A2 AR 241158 A2 AR241158 A2 AR 241158A2 AR 29381583 A AR29381583 A AR 29381583A AR 29381583 A AR29381583 A AR 29381583A AR 241158 A2 AR241158 A2 AR 241158A2
- Authority
- AR
- Argentina
- Prior art keywords
- oxoazetidin
- analogs
- acetic acids
- formula
- yloxy acetic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
- C07D205/085—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a nitrogen atom directly attached in position 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Cephalosporin Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
UN PROCEDIMIENTO PARA PREPARAR BETA-LACTAMAS DE FORMULA (I), Y SUS ESTERES O SALES EN DONDE R1 SIGNIFICA: ENTRE OTROS, (2-AMINO-4-TIAZOLIL)(ALCOXIIMINO)ALCANOILO; (2-AMINO-4-TIAZOLIL)(DIFENILALCOXI)ALQUILOXIALCOXI(IMINO)ALCNOILO; R2 ES H; R3, R4, R5 Y R6 REPRESENTAN H O ALQUILO. EL PROCESO SE BASA EN ACILAR UN COMPUESTO DE FORMULA (II), O SUS ESTERES, CON UN ACIDO DE FORMULA R1-OH, UN HALOGENURO O ANHIDRIDO DEL MISMO, EN DONDE R1 ES UN GRUPO ACILO TAL COMO SE HA DEFINIDO PREVIAMENTE.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US40494582A | 1982-08-04 | 1982-08-04 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AR241158A2 true AR241158A2 (es) | 1991-12-30 |
| AR241158A1 AR241158A1 (es) | 1991-12-30 |
Family
ID=23601669
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AR293815A AR241158A1 (es) | 1982-08-04 | 1983-08-04 | Un procedimiento para la preparacion de compuestos de beta-lactamas y sus sales |
Country Status (33)
| Country | Link |
|---|---|
| US (1) | US4939253A (es) |
| JP (1) | JPS5993046A (es) |
| KR (1) | KR900001211B1 (es) |
| AR (1) | AR241158A1 (es) |
| AT (1) | AT382367B (es) |
| AU (1) | AU568086B2 (es) |
| BE (1) | BE897466A (es) |
| CH (1) | CH655309A5 (es) |
| CS (4) | CS243498B2 (es) |
| DD (1) | DD213919A5 (es) |
| DE (1) | DE3328047A1 (es) |
| DK (1) | DK354683A (es) |
| ES (1) | ES524698A0 (es) |
| FI (1) | FI832675A (es) |
| FR (1) | FR2531427A1 (es) |
| GB (1) | GB2125794B (es) |
| GR (1) | GR79368B (es) |
| HU (1) | HU191058B (es) |
| IE (1) | IE55839B1 (es) |
| IL (1) | IL69381A (es) |
| IN (1) | IN160955B (es) |
| IT (1) | IT1224129B (es) |
| LU (1) | LU84947A1 (es) |
| NL (1) | NL8302746A (es) |
| NO (1) | NO832801L (es) |
| NZ (1) | NZ205111A (es) |
| PL (3) | PL257441A1 (es) |
| PT (1) | PT77155B (es) |
| RO (1) | RO86511B (es) |
| SE (1) | SE8304256L (es) |
| SU (1) | SU1329617A3 (es) |
| YU (1) | YU43324B (es) |
| ZA (1) | ZA835470B (es) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4939253A (en) * | 1982-08-04 | 1990-07-03 | E. R. Squibb & Sons, Inc. | 2-oxoazetidin-1-yloxy acetic acids and analogs |
| US4548747A (en) * | 1983-05-02 | 1985-10-22 | E. R. Squibb & Sons, Inc. | 3-Acylamino-1-sulfonylaminocarbonylmethoxy-2-azetidinones |
| EP0127177B1 (en) * | 1983-05-31 | 1988-12-21 | E.R. Squibb & Sons, Inc. | [[(3-Acylamino-2-oxo-1-azetidinyl)oxy]methyl]phosphinic acids |
| US4534896A (en) * | 1983-06-13 | 1985-08-13 | E. R. Squibb & Sons, Inc. | 3-Acylamino-2-oxoazetidine-1-(β-oxopropionic acid) |
| US4548751A (en) * | 1983-08-03 | 1985-10-22 | E. R. Squibb & Sons, Inc. | (2-Oxo-1-azetidinyloxy)-2-propenoic acid |
| AU581180B2 (en) * | 1983-08-26 | 1989-02-16 | E.R. Squibb & Sons, Inc. | 1-(1h-tetrazol-5-ylalkoxy)-2-azetidinones |
| CA1243679A (en) * | 1983-09-14 | 1988-10-25 | Henner Straub | 3-ACYLAMINO-2-OXO-1-AZETIDINYL-.beta.-OXYPROPIONATES |
| EP0135194A1 (en) * | 1983-09-16 | 1985-03-27 | Takeda Chemical Industries, Ltd. | Azetidinones and their production |
| WO1985004876A1 (en) * | 1984-04-24 | 1985-11-07 | Takeda Chemical Industries, Ltd. | 2-azetidinone derivatives and process for their preparation |
| US4559335A (en) * | 1983-10-03 | 1985-12-17 | E. R. Squibb & Sons, Inc. | 3-Acylamino-1-carboxymethyloxy (or thio) carbonyl-2-azetidinones |
| US4576749A (en) * | 1983-10-03 | 1986-03-18 | E. R. Squibb & Sons, Inc. | 3-Acylamino-1-carboxymethylaminocarbonyl-2-azetidinones |
| US4551277A (en) * | 1983-11-09 | 1985-11-05 | E. R. Squibb & Sons, Inc. | 4-(3-Acylamino-2-oxo-1-azetidinyl)-4-oxo-2-butenoic acid |
| US4581170A (en) * | 1984-08-03 | 1986-04-08 | E. R. Squibb & Sons, Inc. | N-hydroxyl protecting groups and process and intermediates for the preparation of 3-acylamino-1-hydroxy-2-azetidinones |
| EG18314A (en) * | 1985-09-26 | 1993-02-28 | Squibb & Sons Inc | Process for preparing of 2-oxo-1((substituted sulfonyl)amino)carbonyl)-azitidines |
| US5112968A (en) * | 1989-07-28 | 1992-05-12 | E. R. Squibb & Sons, Inc. | Monobactam hydrazide derivatives |
| WO2006055663A2 (en) * | 2004-11-17 | 2006-05-26 | Smithkline Beecham Corporation | The use of novel antibacterial compounds |
| CN102988362B (zh) * | 2005-12-07 | 2014-11-05 | 巴斯利尔药物股份公司 | 单环-内酰胺类抗生素与β-内酰胺酶抑制剂的有效的联合应用 |
| WO2014164526A1 (en) * | 2013-03-13 | 2014-10-09 | Rempex Pharmaceuticals, Inc. | Oxamazin antibiotics |
| US20140275007A1 (en) * | 2013-03-14 | 2014-09-18 | Rempex Pharmaceuticals, Inc. | Oxamazin antibiotics |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ196202A (en) * | 1980-02-07 | 1984-07-31 | Squibb & Sons Inc | Beta-lactam antibiotics (of azetidine-sulphonic acid type) |
| EP0048953B1 (en) * | 1980-09-29 | 1988-03-09 | E.R. Squibb & Sons, Inc. | Beta-lactam antibiotics |
| US4337197A (en) * | 1980-10-31 | 1982-06-29 | E. R. Squibb & Sons, Inc. | O-sulfated β-lactam hydroxamic acids and intermediates |
| WO1982001873A1 (en) * | 1980-12-05 | 1982-06-10 | Takeda Chemical Industries Ltd | 1-sulfo-2-oxoazetidine derivatives and process for their preparation |
| US4939253A (en) * | 1982-08-04 | 1990-07-03 | E. R. Squibb & Sons, Inc. | 2-oxoazetidin-1-yloxy acetic acids and analogs |
-
1983
- 1983-07-21 US US06/515,727 patent/US4939253A/en not_active Expired - Fee Related
- 1983-07-22 FI FI832675A patent/FI832675A/fi not_active Application Discontinuation
- 1983-07-22 HU HU832602A patent/HU191058B/hu not_active IP Right Cessation
- 1983-07-26 ZA ZA835470A patent/ZA835470B/xx unknown
- 1983-07-28 GR GR72076A patent/GR79368B/el unknown
- 1983-07-29 GB GB08320497A patent/GB2125794B/en not_active Expired
- 1983-08-01 IL IL69381A patent/IL69381A/xx unknown
- 1983-08-02 NZ NZ205111A patent/NZ205111A/en unknown
- 1983-08-03 SU SU833635150A patent/SU1329617A3/ru active
- 1983-08-03 AU AU17556/83A patent/AU568086B2/en not_active Ceased
- 1983-08-03 NL NL8302746A patent/NL8302746A/nl unknown
- 1983-08-03 PT PT77155A patent/PT77155B/pt not_active IP Right Cessation
- 1983-08-03 DE DE19833328047 patent/DE3328047A1/de not_active Ceased
- 1983-08-03 SE SE8304256A patent/SE8304256L/xx not_active Application Discontinuation
- 1983-08-03 CS CS85267A patent/CS243498B2/cs unknown
- 1983-08-03 KR KR1019830003626A patent/KR900001211B1/ko not_active IP Right Cessation
- 1983-08-03 ES ES524698A patent/ES524698A0/es active Granted
- 1983-08-03 AT AT0281283A patent/AT382367B/de not_active IP Right Cessation
- 1983-08-03 CS CS85268A patent/CS243499B2/cs unknown
- 1983-08-03 CS CS835759A patent/CS243474B2/cs unknown
- 1983-08-03 IE IE1830/83A patent/IE55839B1/en not_active IP Right Cessation
- 1983-08-03 CS CS83267A patent/CS26783A2/cs unknown
- 1983-08-03 DK DK354683A patent/DK354683A/da not_active Application Discontinuation
- 1983-08-03 NO NO832801A patent/NO832801L/no unknown
- 1983-08-04 PL PL25744183A patent/PL257441A1/xx unknown
- 1983-08-04 AR AR293815A patent/AR241158A1/es active
- 1983-08-04 IT IT22430/83A patent/IT1224129B/it active
- 1983-08-04 FR FR8312862A patent/FR2531427A1/fr active Granted
- 1983-08-04 RO RO111814A patent/RO86511B/ro unknown
- 1983-08-04 PL PL24330883A patent/PL243308A1/xx unknown
- 1983-08-04 BE BE0/211304A patent/BE897466A/fr not_active IP Right Cessation
- 1983-08-04 DD DD83253715A patent/DD213919A5/de not_active IP Right Cessation
- 1983-08-04 LU LU84947A patent/LU84947A1/fr unknown
- 1983-08-04 YU YU1627/83A patent/YU43324B/xx unknown
- 1983-08-04 PL PL25744083A patent/PL257440A1/xx unknown
- 1983-08-04 CH CH4244/83A patent/CH655309A5/fr not_active IP Right Cessation
- 1983-08-04 JP JP58143603A patent/JPS5993046A/ja active Pending
- 1983-08-11 IN IN525/DEL/83A patent/IN160955B/en unknown
Also Published As
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